Novel E3 Ligase Ligand Libraries for Degradation of Proteins Implicated in Malignant Diseases

Authors

  • Béla Bertók ComInnex, Záhony u. 7., H-1031, Budapest, Hungary
  • György Dormán ComInnex, Záhony u. 7., H-1031, Budapest, Hungary
  • Zoltán Várkonyi ComInnex, Záhony u. 7., H-1031, Budapest, Hungary
  • Csaba Magyar Institute of Enzymology, Research Centre for Natural Sciences, Magyar Tudósok Körútja 2., H-1117 Budapest, Hungary

DOI:

https://doi.org/10.33892/aph.2021.91.187-188

Keywords:

PROTAC, protein degradation, E3 ligase binding focused library, cIAP BIR3, 3D virtual screening

Published

2021-11-15

How to Cite

(1)
Bertók, B.; Dormán, G.; Várkonyi, Z.; Magyar, C. Novel E3 Ligase Ligand Libraries for Degradation of Proteins Implicated in Malignant Diseases. Acta Pharm Hung 2021, 91, 187-188.